6ONJ-C-A

PDB Title CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH TRAP220 PEPTIDE AND AGONIST ROSIGLITAZONE
Resolution (Å) 2.300
Classification TRANSCRIPTION/AGONIST

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 259
Binding Area (Å2) 690.65
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.44
Sequence ESADLRALAKHLYDSYIKSFPLTKAKARAILTSPFVIYDMNSLMMGEDKIKHITPLEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1, TRAP220 Coactivator Peptide
Organism Homo sapiens
Chain C
Length 14
Binding Area (Å2) 753.99
Hydrophobic (% a.a.)
42%
Molecular Weight 1668.98
Aromaticity 0.00
Instability -10.29
Isoelectric Point 8.60
Sequence NTKNHPMLMNLLKD

Clustering Classification

Sequence cluster S 184
Contact cluster C8
Interface cluster I1735