3W5R-C-A

PDB Title CRYSTAL STRUCTURE OF COMPLEXES OF VITAMIN D RECEPTOR LIGAND BINDING DOMAIN WITH LITHOCHOLIC ACID DERIVATIVES
Resolution (Å) 2.200
Classification TRANSCRIPTION

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 243
Binding Area (Å2) 515.58
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 5.92
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNEIX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1
Organism Homo sapiens
Chain C
Length 11
Binding Area (Å2) 553.30
Hydrophobic (% a.a.)
54%
Molecular Weight 1338.68
Aromaticity 0.00
Instability -8.10
Isoelectric Point 10.00
Sequence KNHPMLMNLLK

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6