3W0J-C-A

PDB Title CRYSTAL STRUCTURE OF RAT VDR LIGAND BINDING DOMAIN IN COMPLEX WITH NOVEL NONSECOSTEROIDAL LIGANDS
Resolution (Å) 1.840
Classification TRANSCRIPTION

Protein

Description Vitamin D3 Receptor
Organism Rattus norvegicus
Chain A
Length 243
Binding Area (Å2) 495.66
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.21
Sequence RPKLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1
Organism Homo sapiens
Chain C
Length 11
Binding Area (Å2) 539.26
Hydrophobic (% a.a.)
54%
Molecular Weight 1325.60
Aromaticity 0.00
Instability -8.10
Isoelectric Point 6.75
Sequence NHPMLMNLLKD

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6