3VTB-B-A

PDB Title CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR BOUND TO A PARTIAL AGONIST 25-ADAMANTYL-23-YNE-19-NORVITAMMIN D ADTK1
Resolution (Å) 2.000
Classification HORMONE RECEPTOR

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 241
Binding Area (Å2) 517.58
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.06
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description COACTIVATOR PEPTIDE DRIP
Organism -
Chain B
Length 11
Binding Area (Å2) 570.66
Hydrophobic (% a.a.)
54%
Molecular Weight 1338.68
Aromaticity 0.00
Instability -8.10
Isoelectric Point 10.00
Sequence KNHPMLMNLLK

Clustering Classification

Sequence cluster S 184
Contact cluster C1284
Interface cluster I6