3A2H-B-A

PDB Title CRYSTAL STRUCTURE OF THE RAT VITAMIN D RECEPTOR LIGAND BINDING DOMAIN COMPLEXED WITH TEI-9647 AND A SYNTHETIC PEPTIDE CONTAINING THE NR2 BOX OF DRIP 205
Resolution (Å) 2.500
Classification HORMONE RECEPTOR, TRANSCRIPTION

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 240
Binding Area (Å2) 415.05
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 5.92
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNEX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1 peptide
Organism Homo sapiens
Chain B
Length 7
Binding Area (Å2) 472.60
Hydrophobic (% a.a.)
85%
Molecular Weight 831.10
Aromaticity 0.00
Instability -2.20
Isoelectric Point 5.96
Sequence PMLMNLL

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6