3VTC-B-A

PDB Title CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR BOUND TO A PARTIAL AGONIST 26-ADAMANTYL-23-YNE-19-NORVITAMMIN D ADTK3
Resolution (Å) 1.500
Classification HORMONE RECEPTOR

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 241
Binding Area (Å2) 522.20
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.06
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description COACTIVATOR PEPTIDE DRIP
Organism -
Chain B
Length 11
Binding Area (Å2) 588.02
Hydrophobic (% a.a.)
54%
Molecular Weight 1338.68
Aromaticity 0.00
Instability -8.10
Isoelectric Point 10.00
Sequence KNHPMLMNLLK

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6