3W0I-C-A

PDB Title CRYSTAL STRUCTURE OF RAT VDR LIGAND BINDING DOMAIN IN COMPLEX WITH NOVEL NONSECOSTEROIDAL LIGANDS
Resolution (Å) 1.900
Classification TRANSCRIPTION

Protein

Description Vitamin D3 Receptor
Organism Rattus norvegicus
Chain A
Length 243
Binding Area (Å2) 511.01
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.21
Sequence RPKLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1
Organism Homo sapiens
Chain C
Length 12
Binding Area (Å2) 547.92
Hydrophobic (% a.a.)
50%
Molecular Weight 1453.77
Aromaticity 0.00
Instability -6.59
Isoelectric Point 8.60
Sequence KNHPMLMNLLKD

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6