2ZLC-C-A

PDB Title 2-SUBSTITUTED-16-ENE-22-THIA-1ALPHA,25-DIHYDROXY-26,27- DIMETHYL-19-NORVITAMIN D3 ANALOGS: SYNTHESIS, BIOLOGICAL EVALUATION AND CRYSTAL STRUCTURE
Resolution (Å) 2.000
Classification HORMONE

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 241
Binding Area (Å2) 524.34
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.06
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description Coactivator peptide DRIP
Organism -
Chain C
Length 11
Binding Area (Å2) 560.09
Hydrophobic (% a.a.)
54%
Molecular Weight 1338.68
Aromaticity 0.00
Instability -8.10
Isoelectric Point 10.00
Sequence KNHPMLMNLLK

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6