3W0H-C-A

PDB Title CRYSTAL STRUCTURE OF RAT VDR LIGAND BINDING DOMAIN IN COMPLEX WITH NOVEL NONSECOSTEROIDAL LIGANDS
Resolution (Å) 1.800
Classification TRANSCRIPTION

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 248
Binding Area (Å2) 527.37
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.11
Sequence SHDSLRPKLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1
Organism Homo sapiens
Chain C
Length 11
Binding Area (Å2) 563.33
Hydrophobic (% a.a.)
54%
Molecular Weight 1325.60
Aromaticity 0.00
Instability -8.10
Isoelectric Point 6.75
Sequence NHPMLMNLLKD

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6