2ZL9-C-A

PDB Title 2-SUBSTITUTED-16-ENE-22-THIA-1ALPHA,25-DIHYDROXY-26,27- DIMETHYL-19-NORVITAMIN D3 ANALOGS: SYNTHESIS, BIOLOGICAL EVALUATION AND CRYSTAL STRUCTURE
Resolution (Å) 1.900
Classification HORMONE

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 239
Binding Area (Å2) 490.23
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.06
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGX

Peptide

Description Coactivator peptide DRIP
Organism -
Chain C
Length 10
Binding Area (Å2) 526.52
Hydrophobic (% a.a.)
60%
Molecular Weight 1210.51
Aromaticity 0.00
Instability -9.91
Isoelectric Point 8.76
Sequence NHPMLMNLLK

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6