3WT5-C-A

PDB Title A MIXED POPULATION OF ANTAGONIST AND AGONIST BINDING CONFORMERS IN A SINGLE CRYSTAL EXPLAINS PARTIAL AGONISM AGAINST VITAMIN D RECEPTOR: ACTIVE VITAMIN D ANALOGUES WITH 22R-ALKYL GROUP
Resolution (Å) 1.900
Classification TRANSCRIPTION

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 241
Binding Area (Å2) 489.84
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.06
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1
Organism Homo sapiens
Chain C
Length 11
Binding Area (Å2) 533.01
Hydrophobic (% a.a.)
54%
Molecular Weight 1338.68
Aromaticity 0.00
Instability -8.10
Isoelectric Point 10.00
Sequence KNHPMLMNLLK

Clustering Classification

Sequence cluster S 184
Contact cluster C7
Interface cluster I6