6PDZ-C-B

PDB Title CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH SMRT PEPTIDE AND INVERSE AGONIST T0070907
Resolution (Å) 2.100
Classification TRANSCRIPTION

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain B
Length 263
Binding Area (Å2) 446.06
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.48
Sequence QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Nuclear receptor corepressor 2
Organism Homo sapiens
Chain C
Length 13
Binding Area (Å2) 548.47
Hydrophobic (% a.a.)
69%
Molecular Weight 1459.82
Aromaticity 0.00
Instability 9.23
Isoelectric Point 8.75
Sequence NMGLEAIIRKALM

Clustering Classification

Sequence cluster S 198
Contact cluster C8
Interface cluster I1763