5X8Q-D-C

PDB Title CRYSTAL STRUCTURE OF THE MUTANT HUMAN ROR GAMMA LIGAND BINDING DOMAIN WITH ROCKOGENIN.
Resolution (Å) 2.200
Classification TRANSFERASE/IHIBITOR

Protein

Description Nuclear receptor ROR-gamma
Organism Homo sapiens
Chain C
Length 229
Binding Area (Å2) 652.83
Molecular Weight -
Aromaticity 0.09
Instability -
Isoelectric Point 7.19
Sequence SLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPAGKLASLCSQHVERLQIFQHLHPIVX

Peptide

Description Nuclear receptor corepressor 2
Organism Homo sapiens
Chain D
Length 14
Binding Area (Å2) 736.58
Hydrophobic (% a.a.)
71%
Molecular Weight 1516.87
Aromaticity 0.00
Instability 9.29
Isoelectric Point 8.75
Sequence NMGLEAIIRKALMG

Clustering Classification

Sequence cluster S 198
Contact cluster C155
Interface cluster I11