5X8Q-H-G

PDB Title CRYSTAL STRUCTURE OF THE MUTANT HUMAN ROR GAMMA LIGAND BINDING DOMAIN WITH ROCKOGENIN.
Resolution (Å) 2.200
Classification TRANSFERASE/IHIBITOR

Protein

Description Nuclear receptor ROR-gamma
Organism Homo sapiens
Chain G
Length 229
Binding Area (Å2) 692.80
Molecular Weight -
Aromaticity 0.09
Instability -
Isoelectric Point 7.19
Sequence SLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPAGKLASLCSQHVERLQIFQHLHPIVX

Peptide

Description Nuclear receptor corepressor 2
Organism Homo sapiens
Chain H
Length 15
Binding Area (Å2) 754.82
Hydrophobic (% a.a.)
66%
Molecular Weight 1617.97
Aromaticity 0.00
Instability -0.69
Isoelectric Point 8.41
Sequence TNMGLEAIIRKALMG

Clustering Classification

Sequence cluster S 198
Contact cluster C155
Interface cluster I11