6G07-S-D

PDB Title RORGT (264-518;C455S) IN COMPLEX WITH INVERSE AGONIST "CPD-9" AND RIP140 PEPTIDE AT 1.66A
Resolution (Å) 1.660
Classification TRANSCRIPTION

Protein

Description Nuclear receptor ROR-gamma
Organism Homo sapiens
Chain D
Length 246
Binding Area (Å2) 472.80
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 8.19
Sequence YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTX

Peptide

Description Nuclear receptor-interacting protein 1
Organism Homo sapiens
Chain S
Length 10
Binding Area (Å2) 541.43
Hydrophobic (% a.a.)
70%
Molecular Weight 1106.36
Aromaticity 0.00
Instability 33.11
Isoelectric Point 6.71
Sequence VTLLQLLLGH

Clustering Classification

Sequence cluster S 173
Contact cluster C14
Interface cluster I11