3H0A-E-D

PDB Title CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA (PPARG) AND RETINOIC ACID RECEPTOR ALPHA (RXRA) IN COMPLEX WITH 9-CIS RETINOIC ACID, CO-ACTIVATOR PEPTIDE, AND A PARTIAL AGONIST
Resolution (Å) 2.100
Classification TRANSCRIPTION

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain D
Length 266
Binding Area (Å2) 518.31
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.49
Sequence PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Nuclear receptor coactivator 1, Co-activator Peptide
Organism Homo sapiens
Chain E
Length 12
Binding Area (Å2) 570.43
Hydrophobic (% a.a.)
33%
Molecular Weight 1341.55
Aromaticity 0.00
Instability 21.83
Isoelectric Point 8.44
Sequence TSHKLVQLLTTT

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8