2Y0I-S-A

PDB Title FACTOR INHIBITING HIF-1 ALPHA IN COMPLEX WITH TANKYRASE-2 (TNKS2) FRAGMENT PEPTIDE (21-MER)
Resolution (Å) 2.280
Classification OXIDOREDUCTASE/PEPTIDE

Protein

Description HYPOXIA-INDUCIBLE FACTOR 1-ALPHA INHIBITOR
Organism Homo sapiens
Chain A
Length 341
Binding Area (Å2) 796.97
Molecular Weight -
Aromaticity 0.13
Instability -
Isoelectric Point 5.48
Sequence SGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYNXX

Peptide

Description TANKYRASE-2
Organism Homo sapiens
Chain S
Length 14
Binding Area (Å2) 962.38
Hydrophobic (% a.a.)
50%
Molecular Weight 1566.71
Aromaticity 0.07
Instability 13.04
Isoelectric Point 5.14
Sequence SVVEYLLQHGADVH

Clustering Classification

Sequence cluster S 173
Contact cluster C37
Interface cluster I79