6G07-Q-B

PDB Title RORGT (264-518;C455S) IN COMPLEX WITH INVERSE AGONIST "CPD-9" AND RIP140 PEPTIDE AT 1.66A
Resolution (Å) 1.660
Classification TRANSCRIPTION

Protein

Description Nuclear receptor ROR-gamma
Organism Homo sapiens
Chain B
Length 246
Binding Area (Å2) 459.74
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 8.19
Sequence YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTX

Peptide

Description Nuclear receptor-interacting protein 1
Organism Homo sapiens
Chain Q
Length 11
Binding Area (Å2) 510.74
Hydrophobic (% a.a.)
63%
Molecular Weight 1234.53
Aromaticity 0.00
Instability 52.54
Isoelectric Point 8.73
Sequence VTLLQLLLGHK

Clustering Classification

Sequence cluster S 173
Contact cluster C14
Interface cluster I11