6K0T-B-A

PDB Title CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH DIBENZOOXEPINE DERIVATIVE COMPOUND-17
Resolution (Å) 1.840
Classification NUCLEAR PROTEIN

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 262
Binding Area (Å2) 463.25
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.48
Sequence NPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGXQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
Organism Homo sapiens
Chain B
Length 10
Binding Area (Å2) 571.87
Hydrophobic (% a.a.)
70%
Molecular Weight 1095.42
Aromaticity 0.00
Instability 11.28
Isoelectric Point 10.02
Sequence PSLLKKLLLA

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I1689