6AD9-B-A

PDB Title CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH DIBENZOOXEPINE DERIVATIVE COMPOUND-9
Resolution (Å) 2.200
Classification NUCLEAR PROTEIN

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 256
Binding Area (Å2) 470.35
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.62
Sequence SADLRALAKHLYDSYIKSFPLTKAKARAILTGKTDKSPFVIYDMNSLMMGEDKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLX

Peptide

Description 12-mer peptide from Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
Organism Homo sapiens
Chain B
Length 10
Binding Area (Å2) 554.09
Hydrophobic (% a.a.)
70%
Molecular Weight 1095.42
Aromaticity 0.00
Instability 11.28
Isoelectric Point 10.02
Sequence PSLLKKLLLA

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8