5TWO-B-A

PDB Title PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A NOVEL SELECTIVELY PPAR GAMMA-MODULATING LIGAND VSP- 51
Resolution (Å) 1.930
Classification TRANSCRIPTION

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 271
Binding Area (Å2) 466.21
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.75
Sequence ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLX

Peptide

Description PRO-SER-LEU-LEU-LYS-LYS-LEU-LEU-LEU-ALA-PRO
Organism unidentified
Chain B
Length 11
Binding Area (Å2) 560.16
Hydrophobic (% a.a.)
72%
Molecular Weight 1192.53
Aromaticity 0.00
Instability 28.67
Isoelectric Point 10.02
Sequence PSLLKKLLLAP

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8