3V9V-C-A

PDB Title CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR
Resolution (Å) 1.600
Classification TRANSCRIPTION/TRANSCRIPTION REGULATOR

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 259
Binding Area (Å2) 489.34
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.34
Sequence ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Peptide from Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
Organism Homo sapiens
Chain C
Length 11
Binding Area (Å2) 561.46
Hydrophobic (% a.a.)
72%
Molecular Weight 1192.53
Aromaticity 0.00
Instability 28.67
Isoelectric Point 10.02
Sequence PSLLKKLLLAP

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8