1RDT-E-D

PDB Title CRYSTAL STRUCTURE OF A NEW REXINOID BOUND TO THE RXRALPHA LIGAND BINDING DOAMIN IN THE RXRALPHA/PPARGAMMA HETERODIMER
Resolution (Å) 2.400
Classification HORMONE/GROWTH FACTOR

Protein

Description Peroxisome proliferator activated receptor gamma
Organism Homo sapiens
Chain D
Length 254
Binding Area (Å2) 261.04
Molecular Weight -
Aromaticity 0.09
Instability -
Isoelectric Point 5.46
Sequence AESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description LxxLL motif coactivator
Organism Homo sapiens
Chain E
Length 7
Binding Area (Å2) 258.84
Hydrophobic (% a.a.)
42%
Molecular Weight 829.98
Aromaticity 0.00
Instability 69.86
Isoelectric Point 6.00
Sequence KQLSELL

Clustering Classification

Sequence cluster S 122
Contact cluster C668
Interface cluster I8