3B1M-B-A

PDB Title CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR CERCO-A
Resolution (Å) 1.600
Classification TRANSCRIPTION

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 261
Binding Area (Å2) 485.62
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.48
Sequence PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
Organism Homo sapiens
Chain B
Length 11
Binding Area (Å2) 553.29
Hydrophobic (% a.a.)
72%
Molecular Weight 1192.53
Aromaticity 0.00
Instability 28.67
Isoelectric Point 10.02
Sequence PSLLKKLLLAP

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8