6G05-P-A

PDB Title RORGT (264-518;C455S) IN COMPLEX WITH INVERSE AGONIST "CPD-2" AND RIP140 PEPTIDE AT 1.90A
Resolution (Å) 1.900
Classification TRANSCRIPTION

Protein

Description Nuclear receptor ROR-gamma
Organism Homo sapiens
Chain A
Length 246
Binding Area (Å2) 394.75
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 8.19
Sequence YASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLSKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTX

Peptide

Description Nuclear receptor-interacting protein 1
Organism Homo sapiens
Chain P
Length 8
Binding Area (Å2) 472.12
Hydrophobic (% a.a.)
75%
Molecular Weight 870.09
Aromaticity 0.00
Instability 49.50
Isoelectric Point 5.18
Sequence TLLQLLLG

Clustering Classification

Sequence cluster S 173
Contact cluster C1700
Interface cluster I11