3V9T-C-A

PDB Title CRYSTAL STRUCTURE OF THE PPARGAMMA-LBD COMPLEXED WITH A CERCOSPORAMIDE DERIVATIVE MODULATOR
Resolution (Å) 1.650
Classification TRANSCRIPTION/TRANSCRIPTION REGULATOR

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 259
Binding Area (Å2) 491.33
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.63
Sequence PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKISKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETSLHPLLQEIYKDLX

Peptide

Description Peptide from Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
Organism Homo sapiens
Chain C
Length 10
Binding Area (Å2) 565.63
Hydrophobic (% a.a.)
70%
Molecular Weight 1095.42
Aromaticity 0.00
Instability 11.28
Isoelectric Point 10.00
Sequence SLLKKLLLAP

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8