3FUR-H-A

PDB Title CRYSTAL STRUCTURE OF PPARG IN COMPLEX WITH INT131
Resolution (Å) 2.300
Classification TRANSCRIPTION/TRANSCRIPTION REGULATOR

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 258
Binding Area (Å2) 498.15
Molecular Weight -
Aromaticity 0.09
Instability -
Isoelectric Point 5.62
Sequence PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYXX

Peptide

Description Nuclear receptor coactivator 1
Organism synthetic construct
Chain H
Length 12
Binding Area (Å2) 553.99
Hydrophobic (% a.a.)
33%
Molecular Weight 1341.55
Aromaticity 0.00
Instability 21.83
Isoelectric Point 8.44
Sequence TSHKLVQLLTTT

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8