2FVJ-B-A

PDB Title A NOVEL ANTI-ADIPOGENIC PARTIAL AGONIST OF PEROXISOME PROLIFERATOR- ACTIVATED RECEPTOR-GAMMA (PPARG) RECRUITS PPARG-COACTIVATOR-1 ALPHA (PGC1A) BUT POTENTIATES INSULIN SIGNALING IN VITRO
Resolution (Å) 1.990
Classification SIGNALING PROTEIN

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 259
Binding Area (Å2) 480.97
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.48
Sequence ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Nuclear receptor coactivator 1
Organism Homo sapiens
Chain B
Length 10
Binding Area (Å2) 526.08
Hydrophobic (% a.a.)
40%
Molecular Weight 1153.37
Aromaticity 0.00
Instability 24.19
Isoelectric Point 8.76
Sequence HKLVQLLTTT

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I8