6MS7-B-A

PDB Title PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH A NOVEL SELECTIVE PPAR-GAMMA MODULATOR VSP-77
Resolution (Å) 1.430
Classification TRANSCRIPTION

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain A
Length 267
Binding Area (Å2) 476.30
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.49
Sequence GSPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDXX

Peptide

Description PGC1 LXXLL motif
Organism synthetic construct
Chain B
Length 11
Binding Area (Å2) 568.75
Hydrophobic (% a.a.)
72%
Molecular Weight 1192.53
Aromaticity 0.00
Instability 28.67
Isoelectric Point 10.02
Sequence PSLLKKLLLAP

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I1707