2XUM-S-A

PDB Title FACTOR INHIBITING HIF (FIH) Q239H MUTANT IN COMPLEX WITH ZN(II), NOG AND ASP-SUBSTRATE PEPTIDE (20-MER)
Resolution (Å) 2.200
Classification OXIDOREDUCTASE/PEPTIDE

Protein

Description HYPOXIA-INDUCIBLE FACTOR 1-ALPHA INHIBITOR
Organism Homo sapiens
Chain A
Length 351
Binding Area (Å2) 903.53
Molecular Weight -
Aromaticity 0.12
Instability -
Isoelectric Point 5.47
Sequence MAATAAEAVASGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRHSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYNXX

Peptide

Description ASP-SUBSTRATE PEPTIDE 2
Organism synthetic construct
Chain S
Length 18
Binding Area (Å2) 1150.37
Hydrophobic (% a.a.)
50%
Molecular Weight 1979.19
Aromaticity 0.00
Instability -18.62
Isoelectric Point 4.43
Sequence EVVKLLLEHGADVDAQDK

Clustering Classification

Sequence cluster S 173
Contact cluster C37
Interface cluster I79