6K0T-D-C

PDB Title CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH DIBENZOOXEPINE DERIVATIVE COMPOUND-17
Resolution (Å) 1.840
Classification NUCLEAR PROTEIN

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain C
Length 269
Binding Area (Å2) 489.33
Molecular Weight -
Aromaticity 0.09
Instability -
Isoelectric Point 5.92
Sequence NPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPKEVAIRIFQGXQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
Organism Homo sapiens
Chain D
Length 12
Binding Area (Å2) 591.81
Hydrophobic (% a.a.)
58%
Molecular Weight 1353.65
Aromaticity 0.00
Instability 54.28
Isoelectric Point 6.24
Sequence EEPSLLKKLLLA

Clustering Classification

Sequence cluster S 173
Contact cluster C8
Interface cluster I1690