4ZKO-P-U

PDB Title THE CRYSTAL STRUCTURE OF UPAIN-1-W3A IN COMPLEX WITH UPA AT PH7.4
Resolution (Å) 1.290
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 248
Binding Area (Å2) 168.61
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 8.30
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKEX

Peptide

Description N-terminal fragment of upain-1-W3A
Organism synthetic construct
Chain P
Length 2
Binding Area (Å2) 326.56
Hydrophobic (% a.a.)
50%
Molecular Weight 245.28
Aromaticity 0.00
Instability 5.00
Isoelectric Point 9.79
Sequence AR

Clustering Classification

Sequence cluster S 1510
Contact cluster C4
Interface cluster I1322