1EB1-A-H

PDB Title COMPLEX STRUCTURE OF HUMAN THROMBIN WITH N-METHYL-ARGININE INHIBITOR
Resolution (Å) 1.800
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description THROMBIN HEAVY CHAIN
Organism Homo sapiens
Chain H
Length 257
Binding Area (Å2) 480.91
Molecular Weight 29551.69
Aromaticity 0.11
Instability 32.06
Isoelectric Point 8.99
Sequence IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF

Peptide

Description PEPTIDE INHIBITOR
Organism synthetic construct
Chain A
Length 10
Binding Area (Å2) 605.54
Hydrophobic (% a.a.)
50%
Molecular Weight 1209.26
Aromaticity 0.20
Instability 67.82
Isoelectric Point 3.50
Sequence DYEPIPEEAF

Clustering Classification

Sequence cluster S 79
Contact cluster C4
Interface cluster I14