3OX7-P-U

PDB Title THE CRYSTAL STRUCTURE OF UPA COMPLEX WITH PEPTIDE INHIBITOR MH027 AT PH4.6
Resolution (Å) 1.580
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 247
Binding Area (Å2) 573.97
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 8.30
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSALAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKEEX

Peptide

Description MH027
Organism -
Chain P
Length 14
Binding Area (Å2) 805.84
Hydrophobic (% a.a.)
42%
Molecular Weight 1534.74
Aromaticity 0.07
Instability 28.54
Isoelectric Point 6.73
Sequence GACSWRGLENHAMC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I50