3OY5-P-U

PDB Title THE CRYSTAL STRUCTURE OF UPA COMPLEX WITH PEPTIDE INHIBITOR MH027 AT PH7.4
Resolution (Å) 2.310
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 247
Binding Area (Å2) 616.19
Molecular Weight 27822.41
Aromaticity 0.10
Instability 45.16
Isoelectric Point 8.30
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSATLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKEE

Peptide

Description MH027
Organism -
Chain P
Length 15
Binding Area (Å2) 866.85
Hydrophobic (% a.a.)
40%
Molecular Weight 1649.83
Aromaticity 0.07
Instability 27.31
Isoelectric Point 5.32
Sequence DGACSWRGLENHAMC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I50