3OY6-P-U

PDB Title THE CRYSTAL STRUCTURE OF UPA COMPLEX WITH PEPTIDE INHIBITOR MH036 AT PH4.6
Resolution (Å) 2.310
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 247
Binding Area (Å2) 639.43
Molecular Weight 27808.38
Aromaticity 0.10
Instability 42.89
Isoelectric Point 8.30
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE

Peptide

Description MH036
Organism -
Chain P
Length 15
Binding Area (Å2) 863.29
Hydrophobic (% a.a.)
33%
Molecular Weight 1734.94
Aromaticity 0.07
Instability 27.31
Isoelectric Point 6.73
Sequence DGACSWRGLENHRMC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I50