4AX9-I-H

PDB Title HUMAN THROMBIN COMPLEXED WITH NAPSAGATRAN, RO0466240
Resolution (Å) 1.900
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description PROTHROMBIN
Organism Homo sapiens
Chain H
Length 254
Binding Area (Å2) 528.61
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.88
Sequence IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFXXX

Peptide

Description HIRUDIN VARIANT-1
Organism Hirudo medicinalis
Chain I
Length 11
Binding Area (Å2) 595.22
Hydrophobic (% a.a.)
36%
Molecular Weight 1411.47
Aromaticity 0.18
Instability 121.84
Isoelectric Point 3.45
Sequence DFEEIPEEYLQ

Clustering Classification

Sequence cluster S 79
Contact cluster C4
Interface cluster I14