4ZKS-P-U

PDB Title THE CRYSTAL STRUCTURE OF UPAIN-1-W3A IN COMPLEX WITH INACTIVE UPA (UPA-S195A) AT PH7.4
Resolution (Å) 1.850
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 246
Binding Area (Å2) 526.20
Molecular Weight 27663.27
Aromaticity 0.10
Instability 42.24
Isoelectric Point 8.49
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDAGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTK

Peptide

Description upain-1-W3A
Organism synthetic construct
Chain P
Length 12
Binding Area (Å2) 741.93
Hydrophobic (% a.a.)
41%
Molecular Weight 1231.36
Aromaticity 0.00
Instability 38.71
Isoelectric Point 6.73
Sequence CSARGLENHAAC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I50