6XVD-P-U

PDB Title CRYSTAL STRUCTURE OF COMPLEX OF UROKINASE AND A UPAIN-1 VARIANT(W3F) IN PH7.4 CONDITION
Resolution (Å) 1.400
Classification PEPTIDE BINDING PROTEIN

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 248
Binding Area (Å2) 574.55
Molecular Weight 27937.50
Aromaticity 0.10
Instability 44.07
Isoelectric Point 8.05
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKEE

Peptide

Description upain-1-W3F
Organism synthetic construct
Chain P
Length 12
Binding Area (Å2) 810.81
Hydrophobic (% a.a.)
41%
Molecular Weight 1367.58
Aromaticity 0.08
Instability 2.09
Isoelectric Point 6.73
Sequence CSFRGLENHAMC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I1887