3VXE-J-H

PDB Title HUMAN ALPHA-THROMBIN-BIVALIRUDIN COMPLEX AT PD5.0
Resolution (Å) 1.250
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Thrombin heavy chain
Organism Homo sapiens
Chain H
Length 257
Binding Area (Å2) 522.31
Molecular Weight 29551.69
Aromaticity 0.11
Instability 32.06
Isoelectric Point 8.99
Sequence IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF

Peptide

Description BIVALIRUDIN
Organism Hirudo medicinalis
Chain J
Length 10
Binding Area (Å2) 612.54
Hydrophobic (% a.a.)
40%
Molecular Weight 1283.34
Aromaticity 0.20
Instability 100.42
Isoelectric Point 3.45
Sequence DFEEIPEEYL

Clustering Classification

Sequence cluster S 79
Contact cluster C4
Interface cluster I14