4ZHL-P-U

PDB Title THE CRYSTAL STRUCTURE OF MUPAIN-1-IG IN COMPLEX WITH MURINISED HUMAN UPA AT PH7.4
Resolution (Å) 2.060
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 247
Binding Area (Å2) 612.50
Molecular Weight 27834.42
Aromaticity 0.10
Instability 43.73
Isoelectric Point 8.30
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAYHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE

Peptide

Description mupain-1-IG
Organism synthetic construct
Chain P
Length 10
Binding Area (Å2) 856.36
Hydrophobic (% a.a.)
40%
Molecular Weight 1132.31
Aromaticity 0.20
Instability 59.24
Isoelectric Point 8.05
Sequence CPAYSRYIGC

Clustering Classification

Sequence cluster S 329
Contact cluster C4
Interface cluster I50