5WXQ-P-U

PDB Title CRYSTAL STRUCTURE OF UPA IN COMPLEX WITH UPAIN-2-4
Resolution (Å) 1.790
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator chain B
Organism Homo sapiens
Chain U
Length 245
Binding Area (Å2) 601.25
Molecular Weight 27551.10
Aromaticity 0.10
Instability 43.16
Isoelectric Point 8.31
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHT

Peptide

Description upain-2-4 peptide
Organism Phage display vector pTDisp
Chain P
Length 14
Binding Area (Å2) 844.84
Hydrophobic (% a.a.)
42%
Molecular Weight 1474.62
Aromaticity 0.07
Instability 59.93
Isoelectric Point 6.73
Sequence GACSWRGLENHAAC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I50