3M61-P-U

PDB Title CRYSTAL STRUCTURE OF COMPLEX OF UROKINASE AND A UPAIN-1 VARIANT(W3A) IN PH4.6 CONDITION
Resolution (Å) 1.680
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 247
Binding Area (Å2) 553.65
Molecular Weight 27808.38
Aromaticity 0.10
Instability 42.89
Isoelectric Point 8.30
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE

Peptide

Description upain-1 W3A
Organism -
Chain P
Length 12
Binding Area (Å2) 792.96
Hydrophobic (% a.a.)
33%
Molecular Weight 1376.59
Aromaticity 0.00
Instability 2.09
Isoelectric Point 8.08
Sequence CSARGLENHRMC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I50