4X1Q-P-U

PDB Title THE CRYSTAL STRUCTURE OF MUPAIN-1 IN COMPLEX WITH MURINISED HUMAN UPA AT PH7.4
Resolution (Å) 2.280
Classification HYDROLASE INHIBITOR/HYDROLASE

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 247
Binding Area (Å2) 626.35
Molecular Weight 27834.42
Aromaticity 0.10
Instability 43.73
Isoelectric Point 8.30
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADTLAYHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKE

Peptide

Description mupain-1
Organism synthetic construct
Chain P
Length 10
Binding Area (Å2) 849.16
Hydrophobic (% a.a.)
30%
Molecular Weight 1190.35
Aromaticity 0.20
Instability 59.24
Isoelectric Point 5.82
Sequence CPAYSRYLDC

Clustering Classification

Sequence cluster S 329
Contact cluster C4
Interface cluster I50