4ZKN-P-U

PDB Title THE CRYSTAL STRUCTURE OF UPAIN-1-W3A IN COMPLEX WITH UPA AT PH5.5
Resolution (Å) 1.360
Classification HYDROLASE/HYDROLASE INHIBITOR

Protein

Description Urokinase-type plasminogen activator
Organism Homo sapiens
Chain U
Length 247
Binding Area (Å2) 517.71
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 8.49
Sequence IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVYLGRSRLNSNTQGEMKFEVENLILHKDYSADLAHHNDIALLKIRSKEGRCAQPSRTIQTIALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTKMLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPWIRSHTKXX

Peptide

Description upain-1-W3A
Organism synthetic construct
Chain P
Length 12
Binding Area (Å2) 740.59
Hydrophobic (% a.a.)
33%
Molecular Weight 1376.59
Aromaticity 0.00
Instability 2.09
Isoelectric Point 8.08
Sequence CSARGLENHRMC

Clustering Classification

Sequence cluster S 205
Contact cluster C4
Interface cluster I50