6D40-C-A

PDB Title HIGHLY POTENT AND SELECTIVE PLASMIN INHIBITORS BASED ON THE SUNFLOWER TRYPSIN INHIBITOR-1 SCAFFOLD ATTENUATE FIBRINOLYSIS IN PLASMA
Resolution (Å) 1.430
Classification HYDROLASE

Protein

Description Plasminogen
Organism Homo sapiens
Chain A
Length 246
Binding Area (Å2) 543.11
Molecular Weight 26946.72
Aromaticity 0.08
Instability 48.82
Isoelectric Point 8.13
Sequence PSFDCGKPQVEPKKCPVVGGCVAHPHSWPWQVSLRTRFGMHFCGGTLISPEWVLTAAHCLEKSPRPSSYKVILGAHQEVNLEPHVQEIEVSRLFLEPTRKDIALLKLSSPAVITDKVIPACLPSPNYVVADRTECFITGWGETQGTFGAGLLKEAQLPVIENKVCNRYEFLNGRVQSTELCAGHLAGGTDSCQGDSGGPLVCFEKDKYILQGVTSWGLGCARPNKPGVYVRVSRFVTWIEGVMRNN

Peptide

Description Trypsin inhibitor 1
Organism Helianthus annuus
Chain C
Length 14
Binding Area (Å2) 677.94
Hydrophobic (% a.a.)
50%
Molecular Weight 1595.88
Aromaticity 0.14
Instability 29.36
Isoelectric Point 8.05
Sequence GRCYKSIPPICFPD

Clustering Classification

Sequence cluster S 204
Contact cluster C4
Interface cluster I302