2H9T-I-H

PDB Title CRYSTAL STRUCTURE OF HUMAN ALPHA-THROMBIN IN COMPLEX WITH SURAMIN
Resolution (Å) 2.400
Classification HYDROLASE

Protein

Description Thrombin
Organism Homo sapiens
Chain H
Length 251
Binding Area (Å2) 304.10
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.76
Sequence IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGEX

Peptide

Description PPACK active site thrombin inhibitor
Organism -
Chain I
Length 3
Binding Area (Å2) 563.21
Hydrophobic (% a.a.)
66%
Molecular Weight 418.49
Aromaticity 0.33
Instability 45.73
Isoelectric Point 9.75
Sequence FPR

Clustering Classification

Sequence cluster S 143
Contact cluster C4
Interface cluster I46