3HKI-F-E

PDB Title CRYSTAL STRUCTURE OF MURINE THROMBIN MUTANT W215A/E217A IN COMPLEX WITH THE EXTRACELLULAR FRAGMENT OF HUMAN PAR1
Resolution (Å) 2.200
Classification HYDROLASE

Protein

Description Thrombin heavy chain
Organism Mus musculus
Chain E
Length 252
Binding Area (Å2) 491.92
Molecular Weight 29023.27
Aromaticity 0.11
Instability 30.81
Isoelectric Point 9.44
Sequence IVEGWDAEKGIAPWQVMLFRKSPQELLCGASLISDRWVLTAAHCILYPPWDKNFTENDLLVRIGKHSRTRYERNVEKISMLEKIYVHPRYNWRENLDRDIALLKLKKPVPFSDYIHPVCLPDKQTVTSLLRAGYKGRVTGWGNLRETWTNEIQPSVLQVVNLPIVERPVCKASTRIRITDNMFCAGFKVNDTKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSAGAGCGKYGFYTHVFRLKRWIQKVIDQFG

Peptide

Description Proteinase-activated receptor 1
Organism Homo sapiens
Chain F
Length 9
Binding Area (Å2) 625.31
Hydrophobic (% a.a.)
22%
Molecular Weight 1242.29
Aromaticity 0.33
Instability 64.71
Isoelectric Point 4.24
Sequence KYEPFWEDE

Clustering Classification

Sequence cluster S 99
Contact cluster C4
Interface cluster I14