3H0A-B-A

PDB Title CRYSTAL STRUCTURE OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA (PPARG) AND RETINOIC ACID RECEPTOR ALPHA (RXRA) IN COMPLEX WITH 9-CIS RETINOIC ACID, CO-ACTIVATOR PEPTIDE, AND A PARTIAL AGONIST
Resolution (Å) 2.100
Classification TRANSCRIPTION

Protein

Description Retinoic acid receptor RXR-alpha
Organism Homo sapiens
Chain A
Length 211
Binding Area (Å2) 367.75
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 5.82
Sequence EDMPVERILEAELAVENDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLX

Peptide

Description Nuclear receptor coactivator 1, Co-activator Peptide
Organism Homo sapiens
Chain B
Length 11
Binding Area (Å2) 346.53
Hydrophobic (% a.a.)
36%
Molecular Weight 1240.45
Aromaticity 0.00
Instability 22.90
Isoelectric Point 8.44
Sequence TSHKLVQLLTT

Clustering Classification

Sequence cluster S 173
Contact cluster C1168
Interface cluster I9