2ZXN-C-A

PDB Title A NEW CLASS OF VITAMIN D RECEPTOR LIGANDS THAT INDUCE STRUCTURAL REARRANGEMENT OF THE LIGAND-BINDING POCKET
Resolution (Å) 2.100
Classification TRANSCRIPTION

Protein

Description Vitamin D3 receptor
Organism Rattus norvegicus
Chain A
Length 241
Binding Area (Å2) 505.26
Molecular Weight -
Aromaticity 0.07
Instability -
Isoelectric Point 6.06
Sequence KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMSPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNX

Peptide

Description Mediator of RNA polymerase II transcription subunit 1
Organism Xenopus tropicalis
Chain C
Length 11
Binding Area (Å2) 534.07
Hydrophobic (% a.a.)
54%
Molecular Weight 1338.68
Aromaticity 0.00
Instability -8.10
Isoelectric Point 10.00
Sequence KNHPMLMNLLK

Clustering Classification

Sequence cluster S 184
Contact cluster C1091
Interface cluster I6